Monday, August 1, 2022

Complement inhibition in hematologic disease

 


PNH

Loss of CD55 and CD59 due to loss of PIGA coded proteins which bind these proteins using GPI anchors--> alternative pathway for complement activation --> RBC hemolysis.

-C5 inhibitor Ravulizumab

-C3 inhibitor Pegcetacoplan: FDA approved, given subcut twice a week. Main AE infection with encapsulated bacteria. black box warning meningococcal d/s


Cold Agglutinin disease

Ig M binds to RBC and brings along C3b as a companion in lower temp.

 In warmer temp, Ig M dissociates from the RBC, leaving C3b on the RBCs --> hemolysis.

Current rx: avoid cold, rituxan front line, relapsed disease fludarabine rituxan, velcade, BR therapy

-FDA approved sutimlimab--> inhibits classical complement C1

Caution: vaccinate against encapsulated bacteria before starting the treatment.

Initially weekly for 2 doses then every other week.


Transplantation-associated microangiopathy: 

thrombocytopenia, microangiopathic hemolytic anemia, organ damage

Current rx: stop the calcineurin inhibitor, PLEX, rituxan, steroids eculizumab

Lectin pathway and complement inhibition are being investigated in those resistant to eculizumab ( narsoplimab and conversion)


ITP: Sutimlimab being investigated for ITP resistant to prior therapies


Ref: Blood June 2022

No comments:

Post a Comment

Primary CNS lymphoma

 Reference: Annals of Oncology  June 2024 ESMO guidelines Diagnosis  Recommendations • Contrast-enhanced cranial MRI is the recommended imag...